- Article
68Ga-Labeled [Thz14]Bombesin(7–14) Analogs: Promising GRPR-Targeting Agonist PET Tracers with Low Pancreas Uptake
- Lei Wang,
- Ivica Jerolim Bratanovic,
- Zhengxing Zhang,
- Hsiou-Ting Kuo,
- Helen Merkens,
- Jutta Zeisler,
- Chengcheng Zhang,
- Ruiyan Tan,
- François Bénard and
- Kuo-Shyan Lin
With overexpression in various cancers, the gastrin-releasing peptide receptor (GRPR) is a promising target for cancer imaging and therapy. However, the high pancreas uptake of reported GRPR-targeting radioligands limits their clinical application. O...

