- Article
Synthesis and Biological Evaluation of Marine-Inspired Benzothiazole Derivatives as Retinoid X Receptor-α Antagonists with Anti-Cancer Activities
- Yingting Lin,
- Ming Peng,
- Renjing Yang,
- Guanghui Wang,
- Junjie Chen,
- Rong Ding,
- Cuiling Sun,
- Wenjing Tian and
- Haifeng Chen
Retinoid X receptor α (RXRα) plays a vital role in multiple biological and pathological processes and represents a promising therapeutic target for anti-tumor drug design. Inspired by the marine-derived RXRα antagonist meroterpenthi...

