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Topical Advisory Panel for section 'Medicinal Chemistry'

Please see the section webpage for more information on this section.

Members


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Centro de Investigaciones Energéticas, Medioambientales y Tecnológicas (CIEMAT), Madrid, Spain
Interests: pharmacokinetics; radiopharmacy; molecular imaging; PET/CT; radiobiology
Special Issues, Collections and Topics in MDPI journals

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Centro de Química Estrutural, Instituto Superior Técnico, Universidade de Lisboa, 1049-001 Lisboa, Portugal
Interests: adductomics; drug metabolism; mass spectrometry; protein covalent adducts; biomarkers of exposure; diagnosis biomarkers; molecular mechanisms of chemically-induced adverse reactions; bioactivation mechanisms
Special Issues, Collections and Topics in MDPI journals
Department of Pharmacy, University of Salerno, Via Giovanni Paolo II 132, I-84084 Fisciano, Italy
Interests: drug delivery; formulation and modified release; natural polymers; polymer science; particle engineering; pharmaceutical application of micro- and nano-technologies; 3D-printing; polymeric scaffolds for tissue engineering
Special Issues, Collections and Topics in MDPI journals
Department of Cell and Molecular Biology-BMC, Uppsala University, Box 596, SE-751 24 Uppsala, Sweden
Interests: drug design and discovery; molecular recognition; medicinal chemistry; structure-activity relationship; molecular modeling; GPCR; epigenetics; chemical space; virtual screening; cheminformatics
Special Issues, Collections and Topics in MDPI journals
1. Psylo, Sydney, NSW 2000, Australia
2. Faculty of Science, UNSW Sydney, Sydney, NSW 2052, Australia
Interests: organic synthesis; heterocycles; medicinal chemistry; drug discovery; natural products; bioactive compounds; cannabinoids; psychedelics
Laboratory of Forensic Chemistry and Toxicology, National Institute of Legal Medicine and Forensic Sciences, I.P. – South Branch, Rua Manuel Bento de Sousa, n.º 3, 1169-201 Lisboa, Portugal
Interests: method development and validation; hair testing; alternative specimens; drug monitoring; toxicology
Special Issues, Collections and Topics in MDPI journals

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Université de Nantes, Cibles et Médicaments des Infections et du Cancer, IICiMed EA 1155, Département de Chimie Thérapeutique, F-44000 Nantes, France
Interests: medicinal chemistry; organic synthesis; heterocycles; metal-catalyzed cross-coupling reactions; anti-infective agents; anticancer agents
Special Issues, Collections and Topics in MDPI journals

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Institut de Chimie de Nice, UMR CNRS-UNS 7272. Université de Nice Sophia Antipolis. Parc Valrose, 06108 Nice, CEDEX 2, France
Interests: medicinal and green chemistry; chemical biology; targeting resistance in oncology by the design; synthesis and structure-activity relationships of biologically active compounds (small molecules); allosteric inhibitors; validation of new biological targets; targeting RNA and DNA with small molecules; epigenetic and selective stem cells targeting; nucleosides and nucleic acid chemistry


Department of Pharmaceutical Sciences, Wegmans School of Pharmacy, St. John Fisher College, 3690 East Avenue, Room # RCW107, Rochester, NY 14618, USA
Interests: liposomes; targeted drug delivery; niosomes; nanoformulations; PLGA nanoparticles; micelles; thermoreversible gel; controlled release; ocular drug delivery
Special Issues, Collections and Topics in MDPI journals
1. Institute for Research and Innovation in Biomedicine (IRIB), University of Rouen Normandy, LITIS-QUANTIF EA4108, 76000 Rouen, France
2. Department of nuclear medicine, Henri Becquerel Centre, Rouen, France
Interests: radiochemistry; radiopharmacy; nuclear medicine
Special Issues, Collections and Topics in MDPI journals

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Department of Pharmaceutical Technology, Faculty of Pharmacy, University of Debrecen, Nagyerdei körút 98, 4032 Debrecen, Hungary
Interests: assessment of biocompatibility; drug delivery system formulation; application of macromolecules; characterization of dosage forms; in vitro dissolution studies; SEDDS
Special Issues, Collections and Topics in MDPI journals

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CIQUP/Department of Chemistry and Biochemistry, Faculty of Sciences, University of Porto, 4169-007 Porto, Portugal
Interests: medicinal chemistry; organic chemistry; neurodegenerative diseases; infectious diseases
Special Issues, Collections and Topics in MDPI journals

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Department of Physics "Ettore Pancini", University of Naples Federico II, Via Cintia, 80126 Napoli, Italy
Interests: organic chemistry synthesis; carbohydrate chemistry; protein–carbohydrate interaction; protein–peptide interaction; medicinal chemistry; cell biology; cytofluorimetry
Special Issues, Collections and Topics in MDPI journals

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Department of Precision and Regenerative Medicine and Ionian Area, University of Bari Aldo Moro, Bari, Italy
Interests: drug delivery using nanoparticles in vitro; cell imaging; cellular models of inflammation; natural antioxidants for airway epithelium; chronic respiratory diseases
Special Issues, Collections and Topics in MDPI journals

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Department of Clinical Sciences, Faculty of Veterinary Medicine, University of Agricultural Sciences and Veterinary Medicine Cluj-Napoca, 400372 Cluj-Napoca, Romania
Interests: biochemistry and molecular biology; cell biology; veterinary sciences
Special Issues, Collections and Topics in MDPI journals

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UCB, 216 Bath Rd, Slough SL1 3WE, UK
Interests: medicinal chemistry; drug discovery; phenotypic screening; biotransformation; drug metabolism; diabetes; Duchenne muscular dystrophy
Special Issues, Collections and Topics in MDPI journals

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1. Department of Molecular Biology and Genetics, Koc University, Istanbul 34450, Turkey
2. Medicinal and Biological Chemistry Science Farm Joint Research Laboratory, Faculty of Life Sciences, Kumamoto University, Kumamoto, Japan
3. Department of Drug Discovery, Science Farm Ltd., Kumamoto 862-0976, Japan
Interests: computational and medicinal chemistry; multi-target drug design; molecular simulations; drug repositioning; structural biology; target identification; protein-ligand interaction
Special Issues, Collections and Topics in MDPI journals

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CREA—Research Centre for Food and Nutrition, via Ardeatina 546, 00178 Rome, Italy
Interests: molecular biology; bioactive compounds; molecular nutrition; hormone metabolism; cancer; hormone-related diseases; nutrigenomics; nutrigenetics; metabolic disease
Special Issues, Collections and Topics in MDPI journals

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ENSCL École National Supérieure de Chimie de Lille, Villeneuve-d'Ascq, France
Interests: heterocyclic chemistry; natural products (including polyphenols and alcaloids); protein-protein and protein-ligand interactions; antiviral and anticancer agents; the hippo pathway; regenerative medicine
Special Issues, Collections and Topics in MDPI journals
CICS-UBI—Centro de Investigação em Ciências da Saúde, Universidade da Beira Interior, Av. Infante D. Henrique, 6200-506 Covilhã, Portugal
Interests: DNA and RNA G-quadruplexes; G-quadruplexes aptamers; G-quadruplex ligands; biomolecular interactions; biophysical techniques; drug design and development; cancer; drug delivery systems
Special Issues, Collections and Topics in MDPI journals

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Institute of Pharmaceutical Technology and Regulatory Affairs, University of Szeged, H-6720 Szeged, Hungary
Interests: quality by design-based formulation strategies; regulatory science; patient centeredness in dosage form design; alternative administration routes; nose-to-brain delivery
Special Issues, Collections and Topics in MDPI journals

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School of Pharmacy, Concordia University Wisconsin, Mequon, WI, USA
Interests: drug design; opioids; cannabinoids; pain; stress; anxiety; drug abuse; addiction; tolerance; dependence
Department of Physical Pharmacy and Pharmacokinetics, Poznan University of Medical Sciences, 6 Święcickiego St., 60-781 Poznań, Poland
Interests: pharmacokinetics; pharmacogenetics; antiplatelet drugs; pharmacometrics; method validation
Special Issues, Collections and Topics in MDPI journals
Department of Life Science and Biochemical Engineering, Sun Moon University, 70, Sunmoon-ro 221, Tangjeong-myeon, Asan-si, Chungnam 31460, Republic of Korea
Interests: antibiotics; bio-active molecules; nanoparticles; drug development and discovery; chemical biology
Special Issues, Collections and Topics in MDPI journals
European Biomedical Research Institute of Salerno (EBRIS), Via De Renzi, 50, 84125 Salerno, Italy
Interests: NMR spectroscopy; molecular docking; qunatum mechanics; homology modeling; molecular dynamics; drug discovery; configurational and conformational determination
Special Issues, Collections and Topics in MDPI journals

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Institute of Solid State Chemistry and Mechanochemistry, 630090 Novosibirsk, Russia
Interests: mechanochemical preparation of solid dispersions of drugs with excipients in order to increase solubility and reduce the effective dose of drugs; investigation of physicochemical mechanisms for the formation of supramolecular structures of drugs in the mechanochemical pathway for their preparation - intermolecular complexes, self-associates, ve; Investigation of the properties of supramolecular complexes of drugs in solid phases and in aqueous solutions; justification of compositions and ways of synthesis of supramolecular structures of drugs in order to achieve maximum characteristics of bioactivity of drugs; obtaining samples for pharmacological tests and subsequent creation of domestic innovative medicines with increased effectiveness and safety

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School of Pharmacy, Pacific University Oregon, Hillsboro, OR 97123, USA
Interests: drug metabolism; pharmacokinetics; natural products; pharmacodynamics; drug analysis
Special Issues, Collections and Topics in MDPI journals
Molecular Imaging Center Antwerp, University of Antwerp, 2610 Wilrijk, Belgium
Interests: radiochemistry; PET/SPECT imaging; cell death imaging; therapy response evaluation; colorectal cancer

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Istituto per l’Endocrinologia e l’Oncologia Sperimentale del CNR ‘‘G. Salvatore’’, Via S. Pansini 5, 80131 Naples, Italy
Interests: aptamers; cancer; targeted delivery; SELEX
Special Issues, Collections and Topics in MDPI journals
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