- Short Note
N-Benzotriazol-1-yl-methyl-1,2,3,4-tetrahydroisoquinoline
- Cornelia Locher,
- Sara Baldey and
- Naseem Peerzada
Benzotriazole-mediated heteroalkylations have been explored for many synthetic pathways.[...]
January 1999 - 5 articles
Benzotriazole-mediated heteroalkylations have been explored for many synthetic pathways.[...]
We use a method for the calculation of the molecular dipole ( μ ) and quadrupole (θ ) moments and dipole-dipole (α ), dipole-quadrupole ( A) and quadrupole-quadrupole (C ) polarizabilities which we have successfully applied to the benzothiazole (A)-b...
A method to reduce the nitro moiety in dimethyl 4-nitro-4-[1-[2(methoxycarbonyl)ethyl]]heptanedioate using a T-1 Raney nickel catalyst in an acidic environment is reported. The method avoids facile lactam formation.
The inorganic property (I) and organic property (O) values of general organic groups are re-proposed here. Both I and O values of drug and biological molecules or groups can be calculated based on their common group values. The calculation can be per...
Enantiomerically pure, five membered cyclic nitrones, easily obtained in large amounts from protected hydroxyacids and aminoacids such as D- and L-tartaric, L-malic, and L-aspartic acids, give cycloaddition reactions with a good diastereocontrol. The...