Design, Synthesis, and Evaluation of New Anticancer Substances and Radiopharmaceuticals
A special issue of Biomolecules (ISSN 2218-273X). This special issue belongs to the section "Chemical Biology".
Deadline for manuscript submissions: 31 December 2025 | Viewed by 17
Special Issue Editors
Interests: medicinal chemistry; organic synthesis; heterocycles; anticancer activity; antimicrobial activity; SAR
Special Issues, Collections and Topics in MDPI journals
Interests: medicinal chemistry; biomarkers; radiopharmaceuticals; radiomics; anticancer activity; in vitro/in vivo evaluation models; personalized medicine
Special Issues, Collections and Topics in MDPI journals
Special Issue Information
Dear Colleagues,
The development of novel anticancer agents and radiopharmaceuticals remains a multidisciplinary field at the intersection of medicinal chemistry, molecular biology, pharmacology, and nuclear medicine. This research area focuses on the rational design, synthesis, and biological evaluation of new compounds with selective cytotoxicity against cancer cells. A growing emphasis is placed on targeting specific molecular pathways and tumor biomarkers to improve therapeutic efficacy and reduce their systemic toxicity. Radiopharmaceuticals, which combine biologically active molecules with radioactive isotopes, offer both diagnostic and therapeutic (theranostic) potential—enabling personalized treatment strategies and real-time monitoring of therapeutic outcomes. Advances in synthetic methodologies, structure–activity relationship (SAR) studies, and in vitro/in vivo evaluation models are accelerating the translation of promising candidates from bench to bedside. This topic invites contributions highlighting innovative approaches to the design and functional evaluation of small molecules, metal complexes, peptides, or nanoparticles with anticancer and/or radiopharmaceutical applications.
Prof. Dr. Monika Pitucha
Dr. Marta Rusek
Guest Editors
Manuscript Submission Information
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Keywords
- synthesis
- anticancer activity
- radiopharamceuticals
- organic compounds
- medicinal chemistry
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