Radiolabeled Nanoparticles: Molecular Design, Targeting, Therapy, and Imaging
A special issue of Molecules (ISSN 1420-3049). This special issue belongs to the section "Nanochemistry".
Deadline for manuscript submissions: 31 August 2026
Special Issue Editors
Interests: gold nanoparticles; gold naonrods; synthesis and in vivo evaluation
Interests: theranostics; radiolabeling; radiopharmaceuticals; molecular imaging; cancer; radionuclide therapy; radiosynthesis
Special Issues, Collections and Topics in MDPI journals
Special Issue Information
Dear Colleague,
Recently, DDS has attracted attention because it maximizes drug efficacy and minimizes side effects by selectively delivering drugs to diseased areas. Focusing on cancer theranostics, Kratochwil et. al. reported that [225Ac]PSMA-617 showed strong therapeutic effects against metastatic prostate cancer. Watabe et al. disclosed high accumulation and detection of [18F]FAPI-74 to primary and metastatic lesions.
Nanoparticles are also widely used for transporting radionuclides into tumors, e.g., 177Lu-, 225Ac- or 211At-labeled gold nanoparticles for Therapeutics, as well as 99mTc-, 111ln- or 64Cu-labeled liposomes for imaging probes. Additionally, nanoparticles are an excellent tool for drug immobilization; thus, they can be directly administered to the lesion-affected part.
In this Special Issue, we invite researchers who submit innovative research articles related to the synthesis of radiolabeled nanoparticles and its evaluation. The evaluation of nanoparticles includes in vitro and in vivo experiments, such as cytotoxicity, biodistribution, therapeutic effect and imaging tests. The choice of target disease is not limited, but we would appreciate it if there was novelty in the structure and shape of the nanoparticles, as well as be interested in reports on comparisons of biological functions based on their differences.
Dr. Yuichiro Kadonaga
Prof. Dr. Kazuma Ogawa
Guest Editors
Manuscript Submission Information
Manuscripts should be submitted online at www.mdpi.com by registering and logging in to this website. Once you are registered, click here to go to the submission form. Manuscripts can be submitted until the deadline. All submissions that pass pre-check are peer-reviewed. Accepted papers will be published continuously in the journal (as soon as accepted) and will be listed together on the special issue website. Research articles, review articles as well as short communications are invited. For planned papers, a title and short abstract (about 100 words) can be sent to the Editorial Office for announcement on this website.
Submitted manuscripts should not have been published previously, nor be under consideration for publication elsewhere (except conference proceedings papers). All manuscripts are thoroughly refereed through a single-blind peer-review process. A guide for authors and other relevant information for submission of manuscripts is available on the Instructions for Authors page. Molecules is an international peer-reviewed open access semimonthly journal published by MDPI.
Please visit the Instructions for Authors page before submitting a manuscript. The Article Processing Charge (APC) for publication in this open access journal is 2700 CHF (Swiss Francs). Submitted papers should be well formatted and use good English. Authors may use MDPI's English editing service prior to publication or during author revisions.
Keywords
- radiolabeled nanoparticles
- molecular design
- targeting
- therapy
- imaging
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