Enhancing the Bioavailability of Poorly Soluble Drugs
Conflicts of Interest
List of Contributions
- Tedesco, E.; Benetti, F.; Castelli, S.; Fratter, A. Prostatic Therapeutic Efficacy of LENILUTS®, a Novel Formulation with Multi-Active Principles. Pharmaceutics 2022, 14, 1866. https://doi.org/10.3390/pharmaceutics14091866.
- Lee, J.; Lee, J.; Lee, S.; Dinh, L.; Oh, H.; Abuzar, S.; Ahn, J.; Hwang, S. Preparation of Apixaban Solid Dispersion for the Enhancement of Apixaban Solubility and Permeability. Pharmaceutics 2023, 15, 907. https://doi.org/10.3390/pharmaceutics15030907.
- Dharani, S.; Mohamed, E.; Khuroo, T.; Rahman, Z.; Khan, M. Formulation Characterization and Pharmacokinetic Evaluation of Amorphous Solid Dispersions of Dasatinib. Pharmaceutics 2022, 14, 2450. https://doi.org/10.3390/pharmaceutics14112450.
- Xu, Q.; Furuishi, T.; Fukuzawa, K.; Yonemochi, E. Physicochemical Properties and Transdermal Absorption of a Flurbiprofen and Lidocaine Complex in the Non-Crystalline Form. Pharmaceutics 2023, 15, 318. https://doi.org/10.3390/pharmaceutics15020318.
- Abdelkader, A.; Preis, E.; Keck, C. SmartFilm Tablets for Improved Oral Delivery of Poorly Soluble Drugs. Pharmaceutics 2022, 14, 1918. https://doi.org/10.3390/pharmaceutics14091918.
- Zupančič, O.; Doğan, A.; Matić, J.; Kushwah, V.; Alva, C.; Spoerk, M.; Paudel, A. SEDEX—Self-Emulsifying Delivery via Hot Melt Extrusion: A Continuous Pilot-Scale Feasibility Study. Pharmaceutics 2022, 14, 2617. https://doi.org/10.3390/pharmaceutics14122617.
- Choi, S.; Park, E.; Lee, J.; Min, K.; Kim, S.; Jang, D.; Maeng, H.; Jin, S.; Cho, K. Preparation and Characterization of Pazopanib Hydrochloride-Loaded Four-Component Self-Nanoemulsifying Drug Delivery Systems Preconcentrate for Enhanced Solubility and Dissolution. Pharmaceutics 2022, 14, 1875. https://doi.org/10.3390/pharmaceutics14091875.
- Kovačević, M.; German Ilić, I.; Bolko Seljak, K.; Zvonar Pobirk, A. High-Shear Wet Granulation of SMEDDS Based on Mesoporous Carriers for Improved Carvedilol Solubility. Pharmaceutics 2022, 14, 2077. https://doi.org/10.3390/pharmaceutics14102077.
- Mohammadi-Meyabadi, R.; Beirampour, N.; Garrós, N.; Alvarado, H.; Limón, D.; Silva-Abreu, M.; Calpena, A.; Mallandrich, M. Assessing the Solubility of Baricitinib and Drug Uptake in Different Tissues Using Absorption and Fluorescence Spectroscopies. Pharmaceutics 2022, 14, 2714. https://doi.org/10.3390/pharmaceutics14122714.
- He, S.; Mu, H. Microenvironmental pH Modification in Buccal/Sublingual Dosage Forms for Systemic Drug Delivery. Pharmaceutics 2023, 15, 637. https://doi.org/10.3390/pharmaceutics15020637.
- Gadziński, P.; Froelich, A.; Jadach, B.; Wojtyłko, M.; Tatarek, A.; Białek, A.; Krysztofiak, J.; Gackowski, M.; Otto, F.; Osmałek, T. Ionotropic Gelation and Chemical Crosslinking as Methods for Fabrication of Modified-Release Gellan Gum-Based Drug Delivery Systems. Pharmaceutics 2023, 15, 108. https://doi.org/10.3390/pharmaceutics15010108.
- Yu, M.; Liang, M.; An, Q.; Wang, W.; Zhang, B.; Yang, S.; Zhou, J.; Yang, X.; Yang, D.; Zhang, L.; Du, G.; Lu, Y. Versatile Solid Modifications of Multicomponent Pharmaceutical Salts: Novel Metformin–Rhein Salts Based on Advantage Complementary Strategy Design. Pharmaceutics 2023, 15, 1196. https://doi.org/10.3390/pharmaceutics15041196.
- Xiong, T.; Guo, T.; He, Y.; Cao, Z.; Xu, H.; Wu, W.; Wu, L.; Zhu, W.; Zhang, J. Lactone Stabilized by Crosslinked Cyclodextrin Metal-Organic Frameworks to Improve Local Bioavailability of Topotecan in Lung Cancer. Pharmaceutics 2023, 15, 142. https://doi.org/10.3390/pharmaceutics15010142.
- Song, J.; Noh, H.; Lee, S.; Han, H. Lipid/Clay-Based Solid Dispersion Formulation for Improving the Oral Bioavailability of Curcumin. Pharmaceutics 2022, 14, 2269. https://doi.org/10.3390/pharmaceutics14112269.
- Ambrogi, V. A New Challenge for the Old Excipient Calcium Carbonate: To Improve the Dissolution Rate of Poorly Soluble Drugs. Pharmaceutics 2023, 15, 300. https://doi.org/10.3390/pharmaceutics15010300.
- Cysewski, P.; Jeliński, T.; Przybyłek, M.; Nowak, W.; Olczak, M. Solubility Characteristics of Acetaminophen and Phenacetin in Binary Mixtures of Aqueous Organic Solvents: Experimental and Deep Machine Learning Screening of Green Dissolution Media. Pharmaceutics 2022, 14, 2828. https://doi.org/10.3390/pharmaceutics14122828.
- Katona, M.; Nagy-Katona, L.; Szabó, R.; Borbás, E.; Tonka-Nagy, P.; Takács-Novák, K. Multi-Compartmental Dissolution Method, an Efficient Tool for the Development of Enhanced Bioavailability Formulations Containing Poorly Soluble Acidic Drugs. Pharmaceutics 2023, 15, 753. https://doi.org/10.3390/pharmaceutics15030753.
- Homayoonfal, M.; Mousavi, M.; Kiani, H.; Askari, G.; Desobry, S.; Arab-Tehrany, E. Modifying the Stability and Surface Characteristic of Anthocyanin Compounds Incorporated in the Nanoliposome by Chitosan Biopolymer. Pharmaceutics 2022, 14, 1622. https://doi.org/10.3390/pharmaceutics14081622.
- Ruiz-Alcaraz, A.; Núñez-Sánchez, M.; Asensio Ruiz, M.; Martínez-Sánchez, M.; Oliva-Bolarín, A.; Martínez Martínez, T.; Pérez Cuadrado, J.; Ramos-Molina, B.; Lozano-Pérez, A. Optimizing the Preparation of Silk Fibroin Nanoparticles and Their Loading with Polyphenols: Towards a More Efficient Anti-Inflammatory Effect on Macrophages. Pharmaceutics 2023, 15, 263. https://doi.org/10.3390/pharmaceutics15010263.
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Pinal, R. Enhancing the Bioavailability of Poorly Soluble Drugs. Pharmaceutics 2024, 16, 758. https://doi.org/10.3390/pharmaceutics16060758
Pinal R. Enhancing the Bioavailability of Poorly Soluble Drugs. Pharmaceutics. 2024; 16(6):758. https://doi.org/10.3390/pharmaceutics16060758
Chicago/Turabian StylePinal, Rodolfo. 2024. "Enhancing the Bioavailability of Poorly Soluble Drugs" Pharmaceutics 16, no. 6: 758. https://doi.org/10.3390/pharmaceutics16060758
APA StylePinal, R. (2024). Enhancing the Bioavailability of Poorly Soluble Drugs. Pharmaceutics, 16(6), 758. https://doi.org/10.3390/pharmaceutics16060758