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Indolylboronic Acids: Preparation and Applications

Department of Organic Chemistry, University of Chemistry and Technology Prague, Technická 5, 166 28 Prague 6, Czech Republic
Author to whom correspondence should be addressed.
Molecules 2019, 24(19), 3523;
Received: 7 September 2019 / Revised: 24 September 2019 / Accepted: 25 September 2019 / Published: 28 September 2019
(This article belongs to the Special Issue Indole Derivatives: Synthesis and Application)
Indole derivatives are associated with a variety of both biological activities and applications in the field of material chemistry. A number of different strategies for synthesizing substituted indoles by means of the reactions of indolylboronic acids with electrophilic compounds are considered the methods of choice for modifying indoles because indolylboronic acids are easily available, stable, non-toxic and new reactions using indolylboronic acids have been described in the literature. Thus, the aim of this review is to summarize the methods available for the preparation of indolylboronic acids as well as their chemical transformations. The review covers the period 2010–2019. View Full-Text
Keywords: indole; boronic acid; C−H borylation; Suzuki reaction; multicomponent reaction; cross-coupling indole; boronic acid; C−H borylation; Suzuki reaction; multicomponent reaction; cross-coupling
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MDPI and ACS Style

Čubiňák, M.; Edlová, T.; Polák, P.; Tobrman, T. Indolylboronic Acids: Preparation and Applications. Molecules 2019, 24, 3523.

AMA Style

Čubiňák M, Edlová T, Polák P, Tobrman T. Indolylboronic Acids: Preparation and Applications. Molecules. 2019; 24(19):3523.

Chicago/Turabian Style

Čubiňák, Marek, Tereza Edlová, Peter Polák, and Tomáš Tobrman. 2019. "Indolylboronic Acids: Preparation and Applications" Molecules 24, no. 19: 3523.

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