Molecules 2004, 9(7), 527-534; doi:10.3390/90700527
Article

One Step Regioselective Synthesis of 5-Aminoisoxazoles from Nitrile Oxides and α-Cyanoenamines

1,* email, 2 and 1
Received: 26 February 2004; Accepted: 5 April 2004 / Published: 30 June 2004
This is an open access article distributed under the Creative Commons Attribution License which permits unrestricted use, distribution, and reproduction in any medium, provided the original work is properly cited.
Abstract: The 1,3-dipolar cycloaddition of nitrile oxides to 1-cyanoenamines gives 5-aminoisoxazoles regioselectively. Moderate to good yields could be obtained depending on the method used to generate the nitrile oxides. The intermediate isoxazolines could not be isolated.
Keywords: 1-Cyanoenamines; nitrile oxides; 1; 3-dipolar cycloaddition; 5-amino- isoxazoles.
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MDPI and ACS Style

Saad, A.; Vaultier, M.; Derdour, A. One Step Regioselective Synthesis of 5-Aminoisoxazoles from Nitrile Oxides and α-Cyanoenamines. Molecules 2004, 9, 527-534.

AMA Style

Saad A, Vaultier M, Derdour A. One Step Regioselective Synthesis of 5-Aminoisoxazoles from Nitrile Oxides and α-Cyanoenamines. Molecules. 2004; 9(7):527-534.

Chicago/Turabian Style

Saad, Amar; Vaultier, Michel; Derdour, Aïcha. 2004. "One Step Regioselective Synthesis of 5-Aminoisoxazoles from Nitrile Oxides and α-Cyanoenamines." Molecules 9, no. 7: 527-534.

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