Reprint

Novel Approaches for Targeting Metalloproteinases

Edited by
December 2023
214 pages
  • ISBN978-3-0365-9709-6 (Hardback)
  • ISBN978-3-0365-9708-9 (PDF)

This book is a reprint of the Special Issue Novel Approaches for Targeting Metalloproteinases that was published in

Biology & Life Sciences
Chemistry & Materials Science
Medicine & Pharmacology
Summary

This Special Issue is a collection of eleven articles (five reviews and six studies) that describe a wide range of approaches to modulating metalloproteinase activity in disease. The techniques described are in vitro, in vivo, and ex vivo.

Format
  • Hardback
License
© 2022 by the authors; CC BY-NC-ND license
Keywords
carbohydrates; glycoconjugates; MMPs; ADAMs; iminosugars; metzincin inhibitors; matrix metalloproteinases (MMPs), protease; tissue inhibitors of metalloproteinases (TIMPs), exosite; small molecule inhibitors; monoclonal antibodies; proteomics; N-terminomics; terminal amine isotopic labeling of substrates (TAILS); MMP-2; MMP-9; Alzheimer’s disease; AD; neurodegeneration; neuroinflammation; natural compounds; marine compounds; terrestrial compounds; nutraceuticals; Matrix Metalloproteinase inhibitors; bone targeting; bisphosphonates; antitumor agents; skeletal malignancies; osteoarthritis; cartilage; metalloproteinase; targeting; meprin α; meprin β; zinc metalloproteinase; medicinal chemistry; probe development; meprin α; meprin β; zinc metalloproteinase; uHTS; dipeptidyl peptidase III; coumarin derivatives; inhibitor; molecular modeling; metalloproteinase; β-blockers; carvedilol; matrix metalloproteinase-2; ischemia-reperfusion injury; isolated heart perfusion; kidney; obeticholic acid; ischemia/reperfusion; liver; metalloproteinases; MMP-2 inhibitor; cardiac dysfunction; ischemia; n/a