Special Issues

Pharmaceuticals publishes Special Issues to create collections of papers on specific topics, with the aim of building a community of authors and readers to discuss the latest research and develop new ideas and research directions. Special Issues are led by Guest Editors, who are experts on the topic and all Special Issue submissions follow MDPI's standard editorial process. The journal’s Editor-in-Chief and/or designated Editorial Board Member will oversee Guest Editor appointments and Special Issue proposals, checking their content for relevance and ensuring the suitability of the material for the journal. The papers published in a Special Issue will be collected and displayed on a dedicated page of the journal’s website. Further information on MDPI's Special Issue policies and Guest Editor responsibilities can be found here. For any inquiries related to a Special Issue, please contact the Editorial Office.

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Pharmaceutical Formulation Characterization Design, 2nd Edition submission deadline 15 Sep 2026 | 3 articles | Viewed by 3417 | Submission Open
Keywords: Quality by Design; factorial design; design space; solid dosage forms; risk assessment; critical process parameters; quality target product profile
(This special issue belongs to the Section Pharmaceutical Technology)
Structural Insights into Protein Kinases-Targeted Therapies: Overcoming Resistance and Advancing Precision Oncology
edited by David Hecht
submission deadline 20 Sep 2026 | 4 articles | Viewed by 7841 | Submission Open
Keywords: protein kinases inhibitor resistance; structural biology of of protein kinases; computational modeling; drug design; preclinical and clinical studies; precision oncology; ALK resistance for personalized medicine
(This special issue belongs to the Section Medicinal Chemistry)
Natural Antioxidants from Medicinal Plants: Extraction and Bioactivity submission deadline 20 Sep 2026 | 3 articles | Viewed by 2473 | Submission Open
Keywords: natural antioxidants; medicinal plants; extraction methods; bioactivity; phenolic compounds; free radical scavenging; pharmacological potential; in silico and in vitro correlation; molecular modeling
(This special issue belongs to the Section Natural Products)
Computation-Driven Discovery of Modern Small-Molecule Therapeutics: From Enzyme Inhibition to Targeted Protein Degradation submission deadline 20 Sep 2026 | 1 articles | Viewed by 1244 | Submission Open
Keywords: computer-aided drug design; small-molecule drugs; enzyme inhibition; PROTACs; molecular docking; molecular dynamics simulation; artificial intelligence in drug design; virtual screening
(This special issue belongs to the Section AI in Drug Development)
Multiomics Perspective in Pharmacogenomics
edited by
submission deadline 20 Sep 2026 | Viewed by 368 | Submission Open
Keywords: clinical pharmacogenomics; epigenomics in pharmacogenomics; transcriptomics in pharmacogenomics; proteomics and metabolomics in pharmacogenomics; microbiome in pharmacogenomics; multiomics in pharmacogenomics; AI and computational tools in pharmacogenomics; genome profiling in pharmacogenomics; metadata in pharmacogenomics
(This special issue belongs to the Section Pharmacology)
Medicinal Plants: Exploring Plant-Based Bioactive Compounds for Cancer and Metabolic Diseases Prevention and Intervention submission deadline 25 Sep 2026 | 9 articles | Viewed by 27330 | Submission Open
Keywords: cancer; metastasis; tumor growth; tumor spread; bioactive compounds; phytochemicals; medicinal plants; phytochemistry; cancer prevention; cancer intervention; metabolic diseases; metabolism; diabetes; MAFLD; dyslipidemia
(This special issue belongs to the Section Natural Products)
Advances in Prostate Cancer Therapeutics
edited by
submission deadline 25 Sep 2026 | 5 articles | Viewed by 15818 | Submission Open
Keywords: prostate cancer; androgen deprivation therapy (ADT); castration-resistant prostate cancer (CRPC); androgen receptor signaling inhibitors; PARP inhibitors; ionizing radiation therapy; radiopharmaceuticals; immunotherapy; biomarkers; personalized medicine; therapeutic resistance; targeted therapy; combination therapy; hormone-sensitive prostate cancer (HSPC); next-generation therapeutics; translational oncology
(This special issue belongs to the Section Pharmacology)
Heterocyclic Compounds in Medicinal Chemistry, 2nd Edition submission deadline 25 Sep 2026 | 5 articles | Viewed by 14870 | Submission Open
Keywords: heterocycles; drug design; drug discovery; bioactive compounds; structure-based drug design; structure–activity relationship; in silico studies; ADMET properties; multicomponent reactions; phytochemicals
(This special issue belongs to the Section Medicinal Chemistry)
Cutting-Edge Biotechnologies and Applications of Natural Products in Drug R&D and Disease Treatment
edited by
submission deadline 25 Sep 2026 | 4 articles | Viewed by 11142 | Submission Open
Keywords: natural products; bioactive compounds; natural product drug discovery and drug design; natural drug formulation; metabolic engineering for bioactive compounds; natural therapeutic agents; nanoformulations of natural compounds; synthetic biology for natural product biosynthesis; genome editing and creation of novel bioactive compounds
(This special issue belongs to the Section Natural Products)
Natural Products with Anticancer Activity
edited by
submission deadline 25 Sep 2026 | 5 articles | Viewed by 10381 | Submission Open
Keywords: natural products; extracts; anticancer activities; phytochemicals; molecular mechanisms
(This special issue belongs to the Section Medicinal Chemistry)
Natural Products and Bioactive Compounds for the Prevention and Treatment of Non-Communicable Chronic Diseases
edited by
submission deadline 25 Sep 2026 | 5 articles | Viewed by 5344 | Submission Open
Keywords: natural products; phytochemicals; chronic diseases; functional foods; herbal medicine; non-communicable diseases; ethnopharmacology; bioactivity
(This special issue belongs to the Section Natural Products)
Targeting Enzymes in Drug Design and Discovery
edited by
submission deadline 25 Sep 2026 | 3 articles | Viewed by 4316 | Submission Open
Keywords: drug design; computer-aided drug design (CADD); molecular docking; molecular dynamics; QSAR; druggable proteins; synthesis; in vitro and in vivo activity evaluations; ADMET predictions and evaluations
(This special issue belongs to the Section Biopharmaceuticals)
Drug Therapy for Autoimmune and Inflammatory Skin Conditions
edited by Sumatha Channapatna Suresh and Galina Marder
submission deadline 25 Sep 2026 | 2 articles | Viewed by 4114 | Submission Open
Keywords: autoimmune skin disease; psoriasis; immunotherapy; cutaneous lupus; dermatitis; biologic therapies; dermatomyositis; translational therapeutics
(This special issue belongs to the Section Pharmacology)
Advances in the Medicinal Synthesis of Bioactive Compounds submission deadline 25 Sep 2026 | 2 articles | Viewed by 2949 | Submission Open
Keywords: medicinal chemistry; bioactive compounds; synthetic methodologies; structure–activity relationship (SAR); drug discovery; pharmacokinetics; therapeutic agents; green chemistry; computational modeling; interdisciplinary research
(This special issue belongs to the Section Medicinal Chemistry)
Biological Properties of Nanostructures Incorporated in Polymeric Matrices submission deadline 25 Sep 2026 | 2 articles | Viewed by 2667 | Submission Open
Keywords: antimicrobial resistance; cancer; diseases; nanotechnology; polimer
(This special issue belongs to the Section Pharmaceutical Technology)
Drug Delivery Strategies for Brain Targeting and Drug Repurposing: Exploring Alternative Routes and Novel Pharmacological Targets
edited by Paraskevi Papakyriakopoulou and
submission deadline 25 Sep 2026 | 1 articles | Viewed by 2084 | Submission Open
Keywords: drug repurposing; brain drug delivery; delivery-driven repurposing; brain pharmacokinetics; brain pharmacodynamics; CNS-targeted drug delivery
(This special issue belongs to the Section Pharmaceutical Technology)
Fluoroquinolones, 2nd Edition
edited by and
submission deadline 25 Sep 2026 | 1 articles | Viewed by 1498 | Submission Open
Keywords: fluoroquinolones; fluoroquinolone-associated disability; antibiotic safety; fluoroquinolone toxicity; antibiotic stewardship
(This special issue belongs to the Section Pharmacology)
Gut Microbiota Modulation: Probiotics, Postbiotics and Other Bioactive Compounds—2nd Edition submission deadline 25 Sep 2026 | 1 articles | Viewed by 1369 | Submission Open
Keywords: gut microbiota; bioactive compounds; immune system; nutrition respiratory health
Ophthalmic Drugs and Pharmacology
edited by Christin Henein and Sahar Awwad
submission deadline 25 Sep 2026 | 1 articles | Viewed by 1186 | Submission Open
Keywords: ophthalmic diseases; optic neuropathies; eye diseases; glaucoma; corneal disorders; retinal degeneration; ocular surface disease
(This special issue belongs to the Section Pharmacology)
Design and Development of PLGA and Polysaccharide Microparticles submission deadline 25 Sep 2026 | 1 articles | Viewed by 783 | Submission Open
Keywords: drug delivery systems; polymeric systems; nanotechnology; controlled release
(This special issue belongs to the Section Medicinal Chemistry)
Low-Dose Naltrexone for Chronic and Cancer Pain
edited by
submission deadline 25 Sep 2026 | Viewed by 400 | Submission Open
Keywords: low-dose naltrexone; LDN; chronic pain; cancer pain; analgesia; neuroinflammation; endocannabinoid system; pain management
(This special issue belongs to the Section Pharmacology)
Progress of Hydrogel Applications in Novel Drug Delivery Platforms, 2nd Edition submission deadline 25 Sep 2026 | Viewed by 348 | Submission Open
Keywords: hydrogels; targeted drug delivery; drug release; drug delivery; smart hydrogels; stimuli-responsive hydrogels; controlled release; hydrogel-based drug delivery; drug carriers
(This special issue belongs to the Section Pharmaceutical Technology)
Drug Treatment for Ophthalmic Diseases
edited by Doina Gherghel and Stephanie Mroczkowska
submission deadline 25 Sep 2026 | Viewed by 297 | Submission Open
Keywords: novel ocular therapies; drug delivery systems; increased compliance; improved bioavailability; reduced side effects; nanotechnology; gene therapy; artificial intelligence
(This special issue belongs to the Section Pharmacology)
Research Progress in New Drug Discovery Driven by Computational and Experimental Approaches
edited by Sankalp Jain
submission deadline 25 Sep 2026 | Viewed by 283 | Submission Open
Keywords: AI-driven drug discovery; machine learning in drug discovery; computational drug design; virtual screening and experimental validation; integrative computational-experimental approaches
(This special issue belongs to the Section AI in Drug Development)
Impact of Drug Transporter Gene Variation on Pharmacokinetics and Clinical Outcomes in Chronic Disease Therapy submission deadline 28 Sep 2026 | Viewed by 496 | Submission Open
Keywords: drug transporter gene variants; chronic diseases; pharmacokinetics; clinical therapeutic effects; individualized medication; ABCB1; SLC22A family; SLCO1B1
(This special issue belongs to the Section Pharmacology)
Therapeutic Potential of Silver Nanoparticles (AgNPs), 2nd Edition
edited by
submission deadline 30 Sep 2026 | 9 articles | Viewed by 23427 | Submission Open
Keywords: metallic nanostructures; plasmonic nanomaterials; photothermal therapy; photodynamic therapy; antimicrobial; antioxidant; anticancer
(This special issue belongs to the Section Medicinal Chemistry)
Multi-Targeted Natural Products as Therapeutics, 2nd Edition submission deadline 30 Sep 2026 | 7 articles | Viewed by 9660 | Submission Open
Keywords: natural products; medicinal herbs; marine products; animal products; bioactive compounds; multifactorial diseases; multi-targeting phytochemicals
(This special issue belongs to the Section Natural Products)
Neuropharmacology of Plant Extracts and Their Active Compounds (Second Edition) submission deadline 30 Sep 2026 | 5 articles | Viewed by 5685 | Submission Open
Keywords: medicinal plant; mental disorder; preclinical; clinical
(This special issue belongs to the Section Natural Products)
Promising Natural Products with Anti-Inflammatory and Antioxidant Bioactivities: Extraction, Identification, and Biological Evaluation
edited by Sara Vieira and
submission deadline 30 Sep 2026 | 3 articles | Viewed by 5502 | Submission Open
Keywords: bioactive compounds; extraction techniques; anti-inflammatory activity; antioxidant activity; inflammation; inflammatory molecules; signaling pathways
(This special issue belongs to the Section Natural Products)
Targeting Epigenetic Regulation for Cancer Therapy submission deadline 30 Sep 2026 | 2 articles | Viewed by 3408 | Submission Open
Keywords: epigenetics; chromatin remodeling; histone modifications; non-coding RNAs; gene regulation; cancer therapy; epigenetic biomarkers; therapeutic targets
(This special issue belongs to the Section Pharmacology)
Application of 2D and 3D-QSAR Models in Drug Design: 2nd Edition
edited by
submission deadline 30 Sep 2026 | 3 articles | Viewed by 2520 | Submission Open
Keywords: quantitative structure–activity relationship (QSAR); structure–activity relationship (SAR); 3D-QSAR; molecular descriptors; pharmacophore modeling; molecular docking; molecular dynamics; computer-aided drug design (CADD); machine learning in drug discovery; AI-driven drug design
(This special issue belongs to the Section Medicinal Chemistry)
Integrated In Silico, In Cellulo, In Vitro and In Vivo Approaches in Modern Drug Discovery submission deadline 30 Sep 2026 | 1 articles | Viewed by 2086 | Submission Open
Keywords: integrated drug discovery; in silico/in vitro/in cellulo/in vivo studies; multilevel experimental validation; molecular docking; molecular dynamics simulations; QSAR modeling; ADMET prediction; structure–activity relationships (SAR); structure-based drug design; medicinal chemistry; translational pharmacology
(This special issue belongs to the Section Medicinal Chemistry)
Pain Management: Novel Biomarkers and Therapeutic Targets
edited by Lucia Carmela Passacatini and Sara Ilari
submission deadline 30 Sep 2026 | 2 articles | Viewed by 1963 | Submission Open
Keywords: chronic pain; inflammation; oxidative stress; NK cells; immune activation; epigenetic regulation; sirtuins; antioxidants; chronic pain management
(This special issue belongs to the Section Pharmacology)
Advances in Small-Molecule Therapeutics Targeting Signaling Pathways
edited by
submission deadline 30 Sep 2026 | 2 articles | Viewed by 1707 | Submission Open
Keywords: small molecules; natural compounds; synthetic compounds; signaling pathways; drug design; drug development; HTS; computational tools; biological evaluations; QSAR; bioavailability; pharmacokinetics
(This special issue belongs to the Section Medicinal Chemistry)
Integrating Precision Nutrition with Pharmacological Therapies: Mechanisms, Clinical Outcomes, and Therapeutic Efficiency
edited by
submission deadline 30 Sep 2026 | 1 articles | Viewed by 1611 | Submission Open
Keywords: precision nutrition; Foods for Special Medical Purposes (FSMPs); nutritional support; drug–nutrient interactions; pharmacokinetics; pharmacodynamics; personalized medicine; pharmacological therapies; cost-effectiveness; integrated care
(This special issue belongs to the Section Pharmacology)
Nanoplatforms for Enhanced Cancer Therapy
edited by Sang Bong Lee
submission deadline 30 Sep 2026 | 1 articles | Viewed by 1096 | Submission Open
Keywords: nanoplatforms; cancer therapy; cell tracking; molecular imaging; multimodal imaging; radiation therapy; radionuclide therapy; radiotheranostics targeted drug delivery; nanomedicine; tumor targeting; radiosensitization; radioisotope delivery; theranostics; precision oncology
(This special issue belongs to the Section Pharmaceutical Technology)
Natural Compounds as Potential Antibacterial Agents: From Molecular Discovery to Smart Applications
edited by , Altevir Rossato Viana and
submission deadline 30 Sep 2026 | Viewed by 892 | Submission Open
Keywords: natural products; WHO priority pathogens; antimicrobial resistance (AMR); antimicrobial photodynamic inactivation; bioactive compounds; biofilms; smart materials; phytochemicals; drug delivery systems
(This special issue belongs to the Section Natural Products)
Omics Approaches in Drug Discovery, Precision Therapy, and Disease Prevention submission deadline 30 Sep 2026 | 1 articles | Viewed by 891 | Submission Open
Keywords: omics technologies; multi-omics analysis; drug target discovery; biomarker discovery; vaccine target identification; translational therapeutics; genomics; transcriptomics; proteomics; metabolomics; pharmacogenomics
(This special issue belongs to the Section Medicinal Chemistry)
The Therapeutic Potential of Neurotrophin Signaling in Neurodegenerative Disorders
edited by Konstantina Chanoumidou, and
submission deadline 30 Sep 2026 | Viewed by 773 | Submission Open
Keywords: central nervous system; neurodegeneration; neuroinflammation; therapy; neurotrophin receptors; regeneration; myelination
(This special issue belongs to the Section Pharmacology)
Therapeutic Potential of Natural Plant-Derived Compounds in Glioblastoma and Other Brain Tumors submission deadline 30 Sep 2026 | Viewed by 573 | Submission Open
Keywords: glioblastoma; GBM; brain tumors; natural plant‑derived compounds; phytochemicals; blood–brain barrier; signaling targets; tumor microenvironment; therapeutic opportunities; targeted therapy
(This special issue belongs to the Section Natural Products)
Pharmacological Therapies and Biomarkers for Diseases in Correlation with Age Groups of Patients
edited by , Delia Codruta Popa and Stoian Anna-Maria Irina
submission deadline 30 Sep 2026 | Viewed by 549 | Submission Open
Keywords: biomarkers in pediatric diseases; biomarkers in ageing diseases; classical or natural treatments; screening strategies
(This special issue belongs to the Section Pharmacology)
Design, Synthesis and Pharmacological Evaluation of Novel Opioid/Non-Opioid Hybrid Compounds
edited by Justyna Piekielna-Ciesielska and
submission deadline 30 Sep 2026 | Viewed by 373 | Submission Open
Keywords: opioid; opioid hybrids; pain; opioid-related side-effects; tolerance; addiction; neurotransmitters
(This special issue belongs to the Section Medicinal Chemistry)
Spectroscopic and Thermodynamic Insights into Drug-Protein Interactions
edited by Silviya Marcheva Abarova and
submission deadline 30 Sep 2026 | Viewed by 363 | Submission Open
Keywords: drug-protein interaction; circular dichroism spectroscopy; isothermal titration calorimetry; thermodynamic analysis; fluorescence quenching; binding constant; pharmacokinetics; conformational changes; spectroscopic binding assay
(This special issue belongs to the Section Pharmacology)
Membrane Receptors in Disease: Mechanisms and Targeted Therapeutic Strategies submission deadline 30 Sep 2026 | Viewed by 338 | Submission Open
Keywords: membrane receptors; targeted drug; signal transduction; therapeutic antibodies; inhibitor; synthetic
(This special issue belongs to the Section Pharmacology)
Novel Neuroprotective Agents and Therapeutics
edited by Yunna Kim and
submission deadline 30 Sep 2026 | Viewed by 328 | Submission Open
Keywords: neuroprotection; neurodegenerative diseases; neurological disorders; drug discovery; therapeutic development; neuroinflammation; oxidative stress; mitochondrial dysfunction; synaptic plasticity; blood–brain barrier
(This special issue belongs to the Section Pharmacology)
Potential Therapeutic Roles of RNA and Protein Molecules in Cardiovascular Diseases
edited by Wei Zhang
submission deadline 30 Sep 2026 | Viewed by 294 | Submission Open
Keywords: cardiovascular diseases; heart failure; hypercholesterolemia and dyslipidemia; novel therapeutic targets; RNA therapeutics; non-coding RNAs; mRNA therapy; targeted delivery systems; nanomedicine; precision cardiovascular medicine
(This special issue belongs to the Section Biopharmaceuticals)
Management and Treatment of Cardiometabolic Disorders Across the Lifespan
edited by Pasquale Mone, and Luigi Simone Aversa
submission deadline 5 Oct 2026 | 1 articles | Viewed by 912 | Submission Open
Keywords: cardiometabolic disorders; frailty; diabetes; prediabetes; insulin resistance; hypertension; atherosclerotic cardiovascular disease; obesity; metabolic syndrome; plastic surgery
(This special issue belongs to the Section Pharmacology)
Chronic Inflammation: Molecular Mechanisms and Precision Biomarkers
edited by and Raul Patrascu
submission deadline 10 Oct 2026 | 1 articles | Viewed by 1272 | Submission Open
Keywords: chronic inflammation; molecular mechanisms; precision biomarkers; immunopathology; cytokines; tumor microenvironment; head and neck diseases; personalized medicine; inflammatory pathways; translational research
(This special issue belongs to the Section Medicinal Chemistry)
Melatonin Applications in Pharmaceutical Science submission deadline 10 Oct 2026 | Viewed by 634 | Submission Open
Keywords: melatonin; pineal gland; epigenetics; pharmacology; physiology; immunology; pharmaceutics; novel therapies; cancer
(This special issue belongs to the Section Pharmacology)
Natural Pharmacons: Biologically Active Plant-Based Pharmaceuticals—4th Edition submission deadline 15 Oct 2026 | 12 articles | Viewed by 22538 | Submission Open
Keywords: chemical characterization of natural preparations; therapeutic potential of natural matrices in cardiovascular diseases, diabetes, cancer, and neurodegenerative diseases; antimicrobial activity; antioxidant activity; anti-enzymatic activity; anti-inflammatory activity; mechanism of pharmacological actions; structure–activity relationship studies
(This special issue belongs to the Section Natural Products)
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